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5-HT4 antagonist 1

CAS No. 261766-73-8

5-HT4 antagonist 1 ( —— )

产品货号. M26034 CAS No. 261766-73-8

5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥2001 有现货
10MG ¥3013 有现货
25MG ¥5095 有现货
50MG ¥7258 有现货
100MG ¥9882 有现货
500MG ¥19845 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    5-HT4 antagonist 1
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
  • 产品描述
    5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6). (In Vivo):5-HT4 antagonist 1 demonstrates good exposure and prolongs t1/2 in other species with t1/2 of 7, 12, and 21 hours for mice, rats, and mini-pig.
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    Non-cleavable
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    261766-73-8
  • 分子量
    480.6
  • 分子式
    C23H36N4O5S
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    CN1CCN(CC1)S(=O)(=O)CCCN1CCC(CNC(=O)c2cccc3OCCOc23)CC1
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Dale Boger.et al. Chimer containing a targeting portion linked to a scission-activated duocarmycin-type prodrug. WO2009064913A1.
产品手册
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