5-HT4 antagonist 1 ( —— )

产品货号. M26034 CAS No. 261766-73-8

COA

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HPLC

MSDS

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产品名称

5-HT4 antagonist 1
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
产品描述

5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6). (In Vivo):5-HT4 antagonist 1 demonstrates good exposure and prolongs t1/2 in other species with t1/2 of 7, 12, and 21 hours for mice, rats, and mini-pig.
同义词

——
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

Non-cleavable
研究领域

——
适应症

——

1.Dale Boger.et al. Chimer containing a targeting portion linked to a scission-activated duocarmycin-type prodrug. WO2009064913A1.

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